Browse by Publication
![]() | Up a level |
Jump to: Article
Number of items: 22.
Article
Amewu, RichardK;
Chadwick, James;
Hussain, Afthab;
Panda, Somnath;
Rinki, Rinki;
Janneh, Omar;
Ward, StephenA;
Miguel, Candel;
Burrell-Saward, Hollie;
Vivas, Livia;
+1 more...
O'Neill, PaulM;
(2013)
Synthesis and evaluation of the antimalarial, anticancer, and caspase 3 activities of tetraoxane dimers.
Bioorganic & medicinal chemistry, 21 (23).
pp. 7392-7397.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2013.09.047
Full text not available from this repository.
Blackie, MAL;
Beagley, P;
Croft, SL;
Kendrick, H;
Moss, JR;
Chibale, K;
(2007)
Metallocene-based antimalarials: An exploration into the influence of the ferrocenyl moiety on in vitro antimalarial activity in chloroquine-sensitive and chloroquine-resistant strains of Plasmodium falciparum.
Bioorganic & medicinal chemistry, 15 (20).
pp. 6510-6516.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2007.07.012
Full text not available from this repository.
Camps, P;
Duque, MD;
Vázquez, S;
Naesens, L;
Clercq, ED;
Sureda, FX;
López-Querol, M;
Camins, A;
Pallàs, M;
Prathalingam, SR;
+4 more...
Kelly, JM;
Romero, V;
Ivorra, D;
Cortés, D;
(2008)
Synthesis and pharmacological evaluation of several ring-contracted amantadine analogs.
Bioorganic & medicinal chemistry, 16 (23).
pp. 9925-36.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2008.10.028
Full text not available from this repository.
Carrico, D;
Ohkanda, J;
Kendrick, H;
Yokoyama, K;
Blaskovich, MA;
Bucher, CJ;
Buckner, FS;
van Voorhis, WC;
Chakrabarti, D;
Croft, SL;
+3 more...
Gelb, MH;
Sebti, SM;
Hamilton, AD;
(2004)
In vitro and in vivo antimalarial activity of peptidomimetic protein farnesyltransferase inhibitors with improved membrane permeability.
Bioorganic & medicinal chemistry.
p. 6517.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2004.09.020
Full text not available from this repository.
Cottrell, DM;
Capers, J;
Salem, MM;
Deluca-Fradley, K;
Croft, SL;
Werbovetz, KA;
(2004)
Antikinetoplastid activity of 3-aryl-5-thiocyanatomethyl-1,2,4- oxadiazoles.
Bioorganic & medicinal chemistry, 12 (11).
p. 2815.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2004.03.054
Full text not available from this repository.
Daunes, S;
Yardley, V;
Croft, SL;
D'Silva, C;
(2016)
Antiprotozoal glutathione derivatives with flagellar membrane binding activity against T. brucei rhodesiense.
Bioorganic & medicinal chemistry.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2016.12.016
Defaux, J;
Sala, M;
Formosa, X;
Galdeano, C;
Taylor, MC;
Alobaid, WAA;
Kelly, JM;
Wright, CW;
Camps, P;
Munoz-Torrero, D;
(2011)
Huprines as a new family of dual acting trypanocidal-antiplasmodial agents.
Bioorganic & medicinal chemistry, 19 (5).
pp. 1702-1707.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2011.01.028
Duque, MD;
Camps, P;
Profire, L;
Montaner, S;
Vázquez, S;
Sureda, FX;
Mallol, J;
López-Querol, M;
Naesens, L;
De Clercq, E;
+2 more...
Prathalingam, SR;
Kelly, JM;
(2009)
Synthesis and pharmacological evaluation of (2-oxaadamant-1-yl)amines.
Bioorganic & medicinal chemistry, 17 (8).
pp. 3198-206.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2009.02.007
Full text not available from this repository.
Duque, MD;
Camps, P;
Torres, E;
Valverde, E;
Sureda, FX;
Lopez-Querol, M;
Camins, A;
Prathalingam, SR;
Kelly, JM;
Vazquez, S;
(2010)
New oxapolycyclic cage amines with NMDA receptor antagonist and trypanocidal activities.
Bioorganic & medicinal chemistry, 18 (1).
pp. 46-57.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2009.11.017
Full text not available from this repository.
Liu, M;
Wilairat, P;
Croft, SL;
Tan, AL;
Go, ML;
(2003)
Structure-activity relationships of antileishmanial and antimalarial chalcones.
Bioorganic & medicinal chemistry, 11 (13).
pp. 2729-38.
ISSN 0968-0896
DOI: https://doi.org/10.1016/s0968-0896(03)0233-5
Full text not available from this repository.
Liu, M;
Wilairat, P;
Croft, SL;
Tan, ALC;
Go, ML;
(2004)
Structure-activity relationships of antileishmanial and antimalarial chalcones (vol 11, pg 2729, 2003).
Bioorganic & medicinal chemistry, 12 (6).
p. 1569.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2004.01.023
Full text not available from this repository.
Lorente, SO;
Gomez, R;
Jimenez, C;
Cammerer, S;
Yardley, V;
de Luca-Fradley, K;
Croft, SL;
Perez, LMR;
Urbina, J;
Pacanowska, DG;
+1 more...
Gilbert, IH;
(2005)
Biphenylquinuclidines as inhibitors of squalene synthase and growth of parasitic protozoa.
Bioorganic & medicinal chemistry, 13 (10).
pp. 3519-3529.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2005.02.060
Full text not available from this repository.
Lorente, SO;
Jimenez, CJ;
Gros, L;
Yardley, V;
de Luca-Fradley, K;
Croft, SL;
Urbina, JA;
Ruiz-Perez, LM;
Pacanowska, DG;
Gilbert, IH;
(2005)
Preparation of transition-state analogues of sterol 24-methyl transferase as potential anti-parasities.
Bioorganic & medicinal chemistry, 13 (18).
pp. 5435-5453.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2005.06.012
Full text not available from this repository.
Mantyla, A;
Rautio, J;
Nevalainen, T;
Vepsalainen, J;
Juvonen, R;
Kendrick, H;
Garner, T;
Croft, SL;
Jarvinen, T;
(2004)
Synthesis and antileishmanial activity of novel buparvaquone oxime derivatives.
Bioorganic & medicinal chemistry, 12 (13).
p. 3497.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2004.04.032
Full text not available from this repository.
Musonda, CC;
Gut, J;
Rosenthal, PJ;
Yardley, V;
Carvalho de Souza, RC;
Chibale, K;
(2006)
Application of multicomponent reactions to antimalarial drug discovery. Part 2: New antiplasmodial and antitrypanosomal 4-aminoquinoline gamma- and delta-lactams via a 'catch and release' protocol.
Bioorganic & medicinal chemistry, 14 (16).
pp. 5605-15.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2006.04.035
Full text not available from this repository.
Nicoletti, S;
Seifert, K;
Gilbert, IH;
(2010)
Water-soluble polymer-drug conjugates for combination chemotherapy against visceral leishmaniasis.
Bioorganic & medicinal chemistry, 18 (7).
pp. 2559-65.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2010.02.043
Pez, D;
Leal, I;
Zuccotto, F;
Boussard, C;
Brun, R;
Croft, SL;
Yardley, V;
Perez, LMR;
Pacanowska, DG;
Gilbert, IH;
(2003)
2,4-diaminopyrimidines as inhibitors of leishmanial and trypanosomal dihydrofolate reductase.
Bioorganic & medicinal chemistry, 11 (22).
pp. 4693-4711.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2003.08.012
Full text not available from this repository.
Sola, I;
Artigas, A;
Taylor, MC;
Pérez-Areales, FJ;
Viayna, E;
Clos, MV;
Pérez, B;
Wright, CW;
Kelly, JM;
Muñoz-Torrero, D;
(2016)
Synthesis and biological evaluation of N-cyanoalkyl-, N-aminoalkyl-, and N-guanidinoalkyl-substituted 4-aminoquinoline derivatives as potent, selective, brain permeable antitrypanosomal agents.
Bioorganic & medicinal chemistry.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2016.08.036
Sola, I;
Castellà, S;
Viayna, E;
Galdeano, C;
Taylor, MC;
Gbedema, SY;
Pérez, B;
Clos, MV;
Jones, DC;
Fairlamb, AH;
+3 more...
Wright, CW;
Kelly, JM;
Muñoz-Torrero, D;
(2015)
Synthesis, biological profiling and mechanistic studies of 4-aminoquinoline-based heterodimeric compounds with dual trypanocidal-antiplasmodial activity.
Bioorganic & medicinal chemistry, 23 (16).
pp. 5156-67.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2015.01.031
Full text not available from this repository.
Too, K;
Brown, DM;
Bongard, E;
Yardley, V;
Vivas, L;
Loakes, D;
(2007)
Anti-malarial activity of N-6-modified purine analogues.
Bioorganic & medicinal chemistry, 15 (16).
pp. 5551-5562.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2007.05.038
Full text not available from this repository.
Torres, E;
Duque, MD;
Lopez-Querol, M;
Taylor, MC;
Naesens, L;
Ma, CL;
Pinto, LH;
Sureda, FX;
Kelly, JM;
Vazquez, S;
(2012)
Synthesis of benzopolycyclic cage amines: NMDA receptor antagonist, trypanocidal and antiviral activities.
Bioorganic & medicinal chemistry, 20 (2).
pp. 942-948.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2011.11.050
Full text not available from this repository.
Xu, Y;
Cuccui, J;
Denman, C;
Maharjan, T;
Wren, BW;
Wagner, GK;
(2018)
Structure-activity relationships in a new class of non-substrate-like covalent inhibitors of the bacterial glycosyltransferase LgtC.
Bioorganic & medicinal chemistry.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2018.03.006